Discovery of Diaryl Piperidone-Sulfonamide As a Novel Dual-Target Inhibitor of STAT3/CAIX Inducing Ferroptosis in Triple-Negative Breast Cancer Cells

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A series of diaryl piperidone-sulfonamide derivatives were designed as dual inhibitors of STAT3/CAIX and ferroptosis inducers for triple-negative breast cancer
[Journal of Medicinal Chemistry]
AbstractGraphical Abstract