Antibody-Exatecan Conjugates with a Novel Self-Immolative Moiety Overcome Resistance in Colon and Lung Cancer

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The authors designed an antibody-drug conjugates class using a novel self-immolative T moiety for traceless conjugation and release of exatecan, a more potent Topoisomerase I inhibitor with less sensitivity to multidrug resistance.
[Cancer Discovery]
Abstract