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Pulmonary Cell NewsResearchers showed the efficacy of their most potent inhibitors in activating the antitumor response using primary human immune cells from healthy donors.
[Journal of Medicinal Chemistry]
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Muszak, D., Surmiak, E., Plewka, J., Magiera-Mularz, K., Kocik-Krol, J., Musielak, B., Sala, D., Kitel, R., Stec, M., Weglarczyk, K., Siedlar, M., Dömling, A., Skalniak, L., & Holak, T. A. (2021). Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein–Protein Interaction. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.1c00957 Cite
